Definition (MSH)
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Drugs that inhibit cholinesterases. The neurotransmitter ACETYLCHOLINE is rapidly hydrolyzed, and thereby inactivated, by cholinesterases. When cholinesterases are inhibited, the action of endogenously released acetylcholine at cholinergic synapses is potentiated. Cholinesterase inhibitors are widely used clinically for their potentiation of cholinergic inputs to the gastrointestinal tract and urinary bladder, the eye, and skeletal muscles; they are also used for their effects on the heart and the central nervous system.
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Definition (CSP)
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any substance or agent which suppresses, prevents or opposes the action of cholinesterase resulting in the potentiation of the action of endogenously released acetylcholine at cholinergic synapses; cholinesterase inhibition is associated with a variety of acute symptoms such as nausea, vomiting, blurred vision, stomach cramps, and rapid heart rate.
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Concepts |
Pharmacologic Substance
(T121)
, Organic Chemical
(T109)
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MSH |
D002800
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SnomedCT |
52761007, 372765004 |
English |
Agents, Anticholinesterase, Anticholinesterase Agents, Cholinesterase Inhibitors, Inhibitors, Cholinesterase, cholinesterase inhibitor, Anti Cholinesterases, Anti-Cholinesterases, Anticholinesterases, Anticholinesterase Drugs, Drugs, Anticholinesterase, Anticholinest. parasympath., CHOLINESTERASE INHIB, anticholinesterase agents (medication), anticholinesterase agents, Cholinesterase Inhibitor, anticholinesterases, anticholinesterase, anti cholinesterase, cholinesterase inhibitors, Anticholinesterase parasympathomimetics, Cholinesterase inhibitors, Anticholinesterase, Anticholinesterase parasympathomimetic, Cholinesterase inhibitor drug, Anticholinesterase agent (substance), Anticholinesterase agent, Anticholinesterase drug (product), Anticholinesterase drug, Anticholinesterase drug, NOS, Anticholinesterase drug (substance) |
French |
Anticholinestérases, Anti-cholinestérasiques, Anti-cholinestérases, Médicaments anticholinestérasiques, Inhibiteurs de la cholinestérase, Anticholinestérasiques |
Swedish |
Kolinesterashämmare
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Finnish |
Koliiniesteraasin estäjät
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Italian |
Agenti anticolinesterasi, Anticolinesterasi, Farmaci anticolinesterasi, Inibitori della colinesterasi |
Russian |
ANTIKHOLINESTERAZNYE AGENTY, ATSETILKHOLINESTERAZY INGIBITORY, KHOLINESTERAZY INGIBITORY, АНТИХОЛИНЭСТЕРАЗНЫЕ АГЕНТЫ, АЦЕТИЛХОЛИНЭСТЕРАЗЫ ИНГИБИТОРЫ, ХОЛИНЭСТЕРАЗЫ ИНГИБИТОРЫ |
Japanese |
抗コリンエステラーゼ物質, コリンエステラーゼ阻害薬, アセチルコリンエステラーゼ阻害剤, コリンエステラーゼ阻害剤 |
Croatian |
KOLINESTERAZIJSKI INHIBITORI
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Polish |
Inhibitory cholinoesterazy
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Norwegian |
Kolinesterasehemmere
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Czech |
cholinesterasa - inhibitory, inhibitory cholinesteráz |
Spanish |
agente anticolinesterasa (sustancia), agente anticolinesterasa, droga anticolinesterasa (producto), droga anticolinesterasa (sustancia), droga anticolinesterasa, droga inhibidora de la colinesterasa, Agentes Anticolinesterasa, Inhibidores de la Colinesterasa |
German |
Anticholinesterasemittel, Cholinesteraseinhibitoren |
Portuguese |
Agentes Anticolinesterase, Inibidores da Colinesterase |