II. Mechanism
III. Pharmacokinetics
- Converted to Agenerase in vivo
IV. Contraindications
- Sulfonamide Allergy (Exercise caution if used)
V. Adverse Effects
- See Protease Inhibitor for adverse effects attributed to the class
- Perioral Paresthesias
- Rash (19%)
- Severe in some cases
VI. Drug Interactions
- CYP3A4 inhibitor