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Gonadotropin-releasing Hormone Agonist
Aka: Gonadotropin-releasing Hormone Agonist, GnRH agonist, Nafarelin Acetate, Synarel
- Indication
- Endometriosis
- Pathophysiology
- Potentiates Gonadotropin-releasing hormone (GnRH)
- Results in hypoestrogenism or pseudo-Menopause
- Does not cause the same androgenic effects as Danazol
- Dosing: Nafarelin Acetate (Synarel)
- Synarel 200-400 micro-g intranasally bid
- Efficacy
- Effective at regression of lesions and relief of pain
- No proven effect on fertility
- Adverse effects
- Menopausal symptoms
- Hot Flashes
- Insomnia
- Emotional changes
- Bone density loss with prolonged use